WP_MONOAMINE_GPCRS | Return to index | ||||||||
Order | Gene | Description | ref_hepatocyte | HepG2 | HepG2.C3A | HuH.7 | SNU475 | THLE | liver |
1 | ADRA1A | Alpha-1A adrenergic receptor | [1] | -6.04[2] | -1.36[3] | -3.01[4] | -4.96[5] | -5.99[6] | 0.89[7] |
2 | ADRB2 | Beta-2 adrenergic receptor | [8] | -8.06[9] | [10] | [11] | -3.03[12] | -4.37[13] | -2.35[14] |
3 | ADRA1B | Alpha-1B adrenergic receptor | [15] | -8.90[16] | [17] | [18] | -2.55[19] | -2.73[20] | -2.32[21] |
4 | CHRM3 | Muscarinic acetylcholine receptor M3 | [22] | -4.05[23] | 1.29[24] | 2.51[25] | -0.04[26] | -3.52[27] | 0.19[28] |
5 | ADRA2C | Alpha-2C adrenergic receptor | [29] | 3.48[30] | 1.22[31] | 1.18[32] | -2.88[33] | -5.31[34] | -5.78[35] |
6 | HTR1D | 5-hydroxytryptamine receptor 1D | [36] | -2.80[37] | 0.14[38] | -0.36[39] | 1.46[40] | -2.06[41] | -5.92[42] |
7 | HTR2B | 5-hydroxytryptamine receptor 2B | [43] | -2.85[44] | 1.68[45] | -0.43[46] | 3.69[47] | -2.45[48] | 1.19[49] |
8 | HTR7 | 5-hydroxytryptamine receptor 7 | [50] | -2.24[51] | -2.04[52] | -2.89[53] | -0.67[54] | 5.31[55] | -2.69[56] |
9 | DRD4 | D(4) dopamine receptor | [57] | -1.11[58] | 4.26[59] | 2.18[60] | 0.25[61] | -1.68[62] | -3.98[63] |
10 | ADRA1D | Alpha-1D adrenergic receptor | [64] | 0.95[65] | 0.64[66] | -2.36[67] | 4.15[68] | -1.82[69] | -5.66[70] |
11 | HRH1 | Histamine H1 receptor | [71] | -0.74[72] | 3.32[73] | 0.35[74] | 6.70[75] | 6.81[76] | -0.14[77] |
12 | ADRB1 | Beta-1 adrenergic receptor | [78] | -4.61[79] | [80] | 4.22[81] | 0.89[82] | -2.85[83] | -0.39[84] |
13 | DRD5 | D(1B) dopamine receptor | [85] | 1.65[86] | 3.80[87] | 1.05[88] | -2.30[89] | -3.10[90] | -2.09[91] |
14 | CHRM4 | Muscarinic acetylcholine receptor M4 | [92] | 2.42[93] | 3.89[94] | 4.00[95] | -2.03[96] | 1.16[97] | -3.80[98] |
15 | HTR2A | 5-hydroxytryptamine receptor 2A | [99] | [100] | 2.60[101] | [102] | -2.02[103] | -0.28[104] | 2.18[105] |
16 | HRH2 | Histamine H2 receptor | [106] | 1.10[107] | 3.98[108] | -0.30[109] | 1.90[110] | -1.93[111] | 1.96[112] |
17 | ADRA2A | Alpha-2A adrenergic receptor | [113] | -3.69[114] | 1.95[115] | [116] | 1.70[117] | 3.69[118] | 1.44[119] |
18 | HTR4 | 5-hydroxytryptamine receptor 4 | [120] | -2.87[121] | [122] | [123] | [124] | -0.53[125] | 2.33[126] |
19 | HTR1F | 5-hydroxytryptamine receptor 1F | [127] | [128] | [129] | [130] | [131] | [132] | [133] |
20 | HTR1A | 5-hydroxytryptamine receptor 1A | [134] | [135] | [136] | [137] | [138] | [139] | [140] |
21 | DRD2 | D(2) dopamine receptor | [141] | [142] | [143] | [144] | [145] | [146] | [147] |
22 | CHRM2 | Muscarinic acetylcholine receptor M2 | [148] | [149] | [150] | [151] | [152] | [153] | [154] |
23 | HTR2C | 5-hydroxytryptamine receptor 2C | [155] | [156] | [157] | [158] | [159] | [160] | [161] |
24 | HTR5A | 5-hydroxytryptamine receptor 5A | [162] | [163] | [164] | [165] | [166] | [167] | [168] |
25 | HTR1E | 5-hydroxytryptamine receptor 1E | [169] | [170] | [171] | [172] | [173] | [174] | [175] |
26 | DRD3 | D(3) dopamine receptor | [176] | [177] | [178] | [179] | [180] | [181] | [182] |
27 | ADRA2B | Alpha-2B adrenergic receptor | [183] | [184] | [185] | [186] | [187] | [188] | [189] |
28 | HTR6 | 5-hydroxytryptamine receptor 6 | [190] | [191] | [192] | [193] | [194] | [195] | [196] |
29 | CHRM1 | Muscarinic acetylcholine receptor M1 | [197] | [198] | [199] | [200] | [201] | [202] | [203] |
30 | HTR1B | 5-hydroxytryptamine receptor 1B | [204] | [205] | [206] | [207] | [208] | [209] | [210] |
31 | DRD1 | D(1A) dopamine receptor | [211] | [212] | [213] | [214] | [215] | [216] | [217] |
32 | ADRB3 | Beta-3 adrenergic receptor | [218] | [219] | [220] | [221] | [222] | [223] | [224] |
33 | CHRM5 | Muscarinic acetylcholine receptor M5 | [225] | [226] | [227] | [228] | [229] | [230] | [231] |